Research ArticleChemistry
Rapid approach to complex boronic acids
- Constantinos G. Neochoritis1,*,†,
- Shabnam Shaabani1,*,
- Maryam Ahmadianmoghaddam1,
- Tryfon Zarganes-Tzitzikas1,
- Li Gao1,
- Michaela Novotná1,
- Tatiana Mitríková1,
- Atilio Reyes Romero1,
- Marina Ika Irianti1,
- Ruixue Xu1,
- Joe Olechno2,
- Richard Ellson2,
- Victoria Helan3,
- Michael Kossenjans3,
- Matthew R. Groves1 and
- Alexander Dömling1,‡
- 1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
- 2Labcyte Inc., 170 Rose Orchard Way, San Jose, CA 95134, USA.
- 3Hit Discovery, Discovery Sciences, IMED Biotech Unit, AstraZeneca, Mölndal, Gothenburg SE-43183, Sweden.
- ↵‡Corresponding author. Email: a.s.s.domling{at}rug.nl
↵* These authors contributed equally to this work.
† Present address: University of Crete, 70013 Heraklion, Greece.
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Science Advances 05 Jul 2019:
Vol. 5, no. 7, eaaw4607
DOI: 10.1126/sciadv.aaw4607
Vol. 5, no. 7, eaaw4607
DOI: 10.1126/sciadv.aaw4607
Constantinos G. Neochoritis
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Shabnam Shaabani
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Maryam Ahmadianmoghaddam
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Tryfon Zarganes-Tzitzikas
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Li Gao
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Michaela Novotná
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Tatiana Mitríková
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Atilio Reyes Romero
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Marina Ika Irianti
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Ruixue Xu
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Joe Olechno
2Labcyte Inc., 170 Rose Orchard Way, San Jose, CA 95134, USA.
Richard Ellson
2Labcyte Inc., 170 Rose Orchard Way, San Jose, CA 95134, USA.
Victoria Helan
3Hit Discovery, Discovery Sciences, IMED Biotech Unit, AstraZeneca, Mölndal, Gothenburg SE-43183, Sweden.
Michael Kossenjans
3Hit Discovery, Discovery Sciences, IMED Biotech Unit, AstraZeneca, Mölndal, Gothenburg SE-43183, Sweden.
Matthew R. Groves
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
Alexander Dömling
1Pharmacy Department, Drug Design group, University of Groningen, Deusinglaan 1, 9700 AV Groningen, Netherlands.
